In recent years, peptide therapy and bioactive compounds have revolutionised the way we approach aging, weight loss, cognitive function, and overall wellness. Once reserved for elite anti-aging clinics or professional athletes, these compounds are now making their way into mainstream health conversations — and for good reason. From regenerating tissues to improving libido, peptides offer a wide range of benefits that address root causes rather than just symptoms.
In this guide, we explore the standout peptides and bio-compounds categorized by their primary functions — so you can get a bird’s-eye view of how these cutting-edge molecules are reshaping modern medicine and aesthetic as well.
Body Composition & Fat Loss
These peptides and compounds help enhance metabolism, promote fat breakdown, reduce appetite, and support weight loss:
Aminophylline / AOD9604 / Glycyrrhetinic Acid – Promotes localised fat reduction, especially around the waist and thighs.
Tesofensine – Reduces cravings for sweet and fatty foods while improving quality of life.
Tirzepatide Plus – Promotes substantial A1C reductions, appetite control, and cardiometabolic improvements.
Tetradecyl Thioacetic Acid / Amlexanox – Supports fat reduction, lowers LDL cholesterol, and improves insulin resistance.
Methylene Blue – Increases energy and supports metabolic performance.
Skin Health & Anti-Aging
These peptides improve skin elasticity, firmness, and hydration while addressing pigmentation, wrinkles, and sagging:
Copper Tripeptide (GHK-Cu) – Enhances skin structure, reduces wrinkles, heals damaged skin, and reduces hyperpigmentation.
DMAE / Estriol / GHK-Cu / Hyaluronic Acid Biopeptide – Improves hydration, reduces pore size, and rejuvenates aging skin.
GHK-Cu / Argireline / Leuphasyl – Helps reduce facial tension and smooth wrinkles.
GHK-Cu (solo) – Promotes collagen production and protects against UV damage.
Melanotan I – Supports melanin production, enhances tanning, and provides UV protection.
Cognitive Function, Mood & Neurological Health
For those seeking sharper mental focus, emotional balance, or neuroprotection:
FG LOOP (FGL) – Enhances mood, cognitive clarity, and neuroplasticity.
Pinealon – Offers neuroprotection, supports cognitive enhancement, and improves sleep.
Synapsin – Improves memory, reduces brain inflammation, and enhances mental acuity.
NAD+ – Revitalizes cellular energy and supports neurological recovery.
Methylene Blue – Improves mood, focus, and mitochondrial function.
SS-31 (Elamipretide) – Offers neuroprotection and addresses neurodegenerative conditions.
Injury Repair, Recovery & Regeneration
These peptides support rapid healing from injuries and optimize recovery:
Pentadeca Arginate – Accelerates healing of tendons, wounds, and bones.
TB-500 – Enhances tissue repair, reduces scar formation, and increases stamina.
Sermorelin – Boosts natural growth hormone release for muscle recovery and body composition improvements.
Thymulin – Supports immune modulation and reduces inflammatory responses.
GHK-Cu – Promotes wound healing and tissue regeneration.
Sexual Health & Libido
Optimized sexual wellness for both men and women:
PT-141 (Bremelanotide) – Enhances sexual desire and treats hypoactive sexual desire disorder in both sexes.
Sermorelin – Improves libido and overall sense of well-being.
Longevity, Detox & Anti-Aging
These compounds focus on cellular health, detoxification, and age-related disease prevention:
NAD+ – Supports cellular repair, detoxification, and mitochondrial function.
Sirolimus – Known for its potential in lifespan extension and prevention of age-related diseases.
SS-31 (Elamipretide) – Protects mitochondrial health and is studied for anti-aging effects.
VIP (Vasoactive Intestinal Peptide) – Beneficial for mold illness and brain healing.
Thymulin – Supports immune resilience in aging individuals.
Why Peptides Are the Future of Functional Health
What makes peptides and bioactive compounds so powerful is their precision. Unlike many traditional medications that mask symptoms, peptides often go straight to the root — activating your body’s own healing and regulatory systems. They’re small in size but mighty in impact, capable of initiating cascades of regeneration, fat-burning, mood balance, or cellular repair.
With continued research, the applications of these molecules continue to expand — from helping people recover faster after injuries to improving skin at the cellular level, enhancing mental clarity, and even reversing signs of aging.
Final Thoughts
Peptide therapy represents the convergence of science, aesthetics, and functional medicine. Whether your goal is to improve your skin, lose stubborn weight, boost your mood, or heal from chronic conditions, there is likely a peptide that can support your journey.
As always, it’s critical to work with a qualified healthcare provider who is an expert in this area to determine the best therapeutic option based on your unique needs. But one thing is clear: the era of personalised medicine powered by peptides is here, and it’s only just a beginning.